Assay Detail
Binding
CHEMBL3624414
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Inhibition of glycogen phosphorylase (unknown origin)
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Computationally motivated synthesis and enzyme kinetic evaluation of N-(-d-glucopyranosyl)-1,2,4-triazolecarboxamides as glycogen phosphorylase inhibitors
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 3 | 6.63 | 6.80 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL490175 | — | — | 1 | 6.80 |
| CHEMBL490001 | — | — | 1 | 6.46 |
| CHEMBL423707 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL490175 | — | Ki | = | 160.0 | nM | 6.80 |
| CHEMBL490001 | — | Ki | = | 350.0 | nM | 6.46 |
| CHEMBL423707 | — | Ki | = | 1700000.0 | nM | - |