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Assay Detail

CHEMBL3626556

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Binding
Inhibition of Vibrio cholerae alpha-carbonic anhydrase by [18O]-exchange mass spectroscopy
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Vibrio cholerae
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

Unchecked (CHEMBL612545)
Type UNCHECKED

Publication

Activity and anion inhibition studies of the α-carbonic anhydrase from Thiomicrospira crunogena XCL-2 Gammaproteobacterium.
Mahon BP, Díaz-Torres NA, Pinard MA, Tu C, Silverman DN, Scott KM, McKenna R.
Bioorg Med Chem Lett (2015) 25 : 4937 -4940
PubMed 25998503 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 4 4.13 4.13

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1200739 HYDROGEN SULFIDE 1 4.13
CHEMBL1231821 HYDROCHLORIC ACID -1.0 1 -
CHEMBL1231461 BROMIDE 1 -
CHEMBL1233550 IODIDE -1.0 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1200739 HYDROGEN SULFIDE Ki = 74000.0 nM 4.13
CHEMBL1231821 HYDROCHLORIC ACID Ki = 930000.0 nM -
CHEMBL1231461 BROMIDE Ki = 28000000.0 nM -
CHEMBL1233550 IODIDE Ki = 9730000.0 nM -