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Assay Detail

CHEMBL3626588

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Binding affinity to human CBP by ITC analysis
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

CREB-binding protein (CHEMBL5747)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Strategies for the Discovery of Target-Specific or Isoform-Selective Modulators.
Zhan P, Itoh Y, Suzuki T, Liu X.
J Med Chem (2015) 58 : 7611 -7633
PubMed 26086931 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Kd 1 7.68 7.68

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL3622373 1 7.68

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL3622373 Kd = 21.0 nM 7.68