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Assay Detail

CHEMBL3635189

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Physicochemical
Metal chelating activity assessed as inhibition of Fe2+-ferrozine complex formation after 10 mins
5
Total Activities
5
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Physicochemical
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Publication

Identification of Highly Promising Antioxidants/Neuroprotectants Based on Nucleoside 5'-Phosphorothioate Scaffold. Synthesis, Activity, and Mechanisms of Action.
Azran S, Danino O, Förster D, Kenigsberg S, Reiser G, Dixit M, Singh V, Major DT, Fischer B.
J Med Chem (2015) 58 : 8427 -8443
PubMed 26447940 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 5 4.06 4.07

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL335206 1 4.07
CHEMBL780 PENTETIC ACID 4.0 1 4.05
CHEMBL14830 ADENOSINE DIPHOSPHATE 0.5 1 -
CHEMBL153 TROLOX 1 -
CHEMBL1261 CITRIC ACID 4.0 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL335206 IC50 = 85000.0 nM 4.07
CHEMBL780 PENTETIC ACID IC50 = 90000.0 nM 4.05
CHEMBL14830 ADENOSINE DIPHOSPHATE IC50 = 250000.0 nM -
CHEMBL153 TROLOX IC50 = 150000.0 nM -
CHEMBL1261 CITRIC ACID IC50 = 300000.0 nM -