Assay Detail
Binding
CHEMBL3720980
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of N-terminal Flag-tagged mouse TRPM7 expressed in HEK293T cells assessed as reduction in whole cell currents by whole-cell patch clamp assay
14
Total Activities
14
Compounds Tested
2
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Mus musculus |
| Cell Type | HEK-293T |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Transient receptor potential cation channel subfamily M member 7 (CHEMBL3714706) ↗| Type | SINGLE PROTEIN |
| Organism | Mus musculus |
Publication
Agents and methods for treating ischemic and other diseases
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| INH | 13 | - | - |
| IC50 | 1 | 5.30 | 5.30 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3716072 | — | — | 1 | 5.30 |
| CHEMBL3717981 | — | — | 1 | - |
| CHEMBL3718897 | — | — | 1 | - |
| CHEMBL3719019 | — | — | 1 | - |
| CHEMBL3716025 | — | — | 1 | - |
| CHEMBL3714873 | — | — | 1 | - |
| CHEMBL3715764 | — | — | 1 | - |
| CHEMBL3715537 | — | — | 1 | - |
| CHEMBL3716221 | — | — | 1 | - |
| CHEMBL3718551 | — | — | 1 | - |
| CHEMBL3717076 | — | — | 1 | - |
| CHEMBL3717768 | — | — | 1 | - |
| CHEMBL3718974 | — | — | 1 | - |
| CHEMBL3718703 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3716072 | — | IC50 | = | 5000.0 | nM | 5.30 |
| CHEMBL3717981 | — | INH | = | 5.0 | uM | - |
| CHEMBL3718897 | — | INH | = | 5.0 | uM | - |
| CHEMBL3719019 | — | INH | = | 5.0 | uM | - |
| CHEMBL3716025 | — | INH | = | 5.0 | uM | - |
| CHEMBL3714873 | — | INH | = | 5.0 | uM | - |
| CHEMBL3715764 | — | INH | = | 5.0 | uM | - |
| CHEMBL3715537 | — | INH | = | 5.0 | uM | - |
| CHEMBL3716221 | — | INH | = | 5.0 | uM | - |
| CHEMBL3718551 | — | INH | = | 5.0 | uM | - |
| CHEMBL3717076 | — | INH | = | 5.0 | uM | - |
| CHEMBL3717768 | — | INH | = | 5.0 | uM | - |
| CHEMBL3718974 | — | INH | = | 5.0 | uM | - |
| CHEMBL3718703 | — | INH | = | 5.0 | uM | - |