Assay Detail
Functional
CHEMBL3734080
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of CRAC in rat RBL2H3 cells assessed as interacellular calcium level after 30 mins by FLIPR assay
71
Total Activities
71
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Rattus norvegicus |
| Cell Type | RBL-2H3 |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Calcium release-activated calcium channel protein 1 (CHEMBL3721308) ↗| Type | SINGLE PROTEIN |
| Organism | Rattus norvegicus |
Publication
Compounds that modulate intracellular calcium
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 71 | 6.22 | 6.22 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3731997 | — | — | 1 | 6.22 |
| CHEMBL3728717 | — | — | 1 | 6.22 |
| CHEMBL3727759 | — | — | 1 | 6.22 |
| CHEMBL3731071 | — | — | 1 | 6.22 |
| CHEMBL3732485 | — | — | 1 | 6.22 |
| CHEMBL3728472 | — | — | 1 | - |
| CHEMBL3729327 | — | — | 1 | - |
| CHEMBL3732098 | — | — | 1 | - |
| CHEMBL3733011 | — | — | 1 | - |
| CHEMBL3728924 | — | — | 1 | - |
| CHEMBL3732872 | — | — | 1 | - |
| CHEMBL3729608 | — | — | 1 | - |
| CHEMBL3729622 | — | — | 1 | - |
| CHEMBL3727596 | — | — | 1 | - |
| CHEMBL3728373 | — | — | 1 | - |
| CHEMBL3730994 | — | — | 1 | - |
| CHEMBL3727582 | — | — | 1 | - |
| CHEMBL3733297 | — | — | 1 | - |
| CHEMBL3728084 | — | — | 1 | - |
| CHEMBL3729876 | — | — | 1 | - |
| CHEMBL3732833 | — | — | 1 | - |
| CHEMBL3731260 | — | — | 1 | - |
| CHEMBL3731335 | — | — | 1 | - |
| CHEMBL3730751 | — | — | 1 | - |
| CHEMBL3729573 | — | — | 1 | - |
| CHEMBL3732454 | — | — | 1 | - |
| CHEMBL3732851 | — | — | 1 | - |
| CHEMBL3729364 | — | — | 1 | - |
| CHEMBL3729028 | — | — | 1 | - |
| CHEMBL3732550 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3731997 | — | IC50 | = | 600.0 | nM | 6.22 |
| CHEMBL3728717 | — | IC50 | = | 600.0 | nM | 6.22 |
| CHEMBL3727759 | — | IC50 | = | 600.0 | nM | 6.22 |
| CHEMBL3731071 | — | IC50 | = | 600.0 | nM | 6.22 |
| CHEMBL3732485 | — | IC50 | = | 600.0 | nM | 6.22 |
| CHEMBL3727582 | — | IC50 | < | 600.0 | nM | - |
| CHEMBL3730725 | — | IC50 | < | 600.0 | nM | - |
| CHEMBL3729327 | — | IC50 | < | 600.0 | nM | - |
| CHEMBL3730095 | — | IC50 | < | 600.0 | nM | - |
| CHEMBL3731956 | — | IC50 | < | 600.0 | nM | - |
| CHEMBL3733351 | — | IC50 | < | 600.0 | nM | - |
| CHEMBL3727392 | — | IC50 | < | 600.0 | nM | - |
| CHEMBL3727719 | — | IC50 | < | 600.0 | nM | - |
| CHEMBL3730577 | — | IC50 | < | 600.0 | nM | - |
| CHEMBL3727557 | — | IC50 | < | 600.0 | nM | - |
| CHEMBL3732356 | — | IC50 | < | 600.0 | nM | - |
| CHEMBL3733096 | — | IC50 | < | 600.0 | nM | - |
| CHEMBL3732172 | — | IC50 | < | 600.0 | nM | - |
| CHEMBL3732517 | — | IC50 | < | 600.0 | nM | - |
| CHEMBL3728586 | — | IC50 | < | 600.0 | nM | - |
| CHEMBL3728333 | — | IC50 | < | 600.0 | nM | - |
| CHEMBL3730066 | — | IC50 | < | 600.0 | nM | - |
| CHEMBL3730763 | — | IC50 | < | 600.0 | nM | - |
| CHEMBL3727650 | — | IC50 | < | 600.0 | nM | - |
| CHEMBL3728688 | — | IC50 | < | 600.0 | nM | - |
| CHEMBL3733110 | — | IC50 | < | 600.0 | nM | - |
| CHEMBL3731436 | — | IC50 | < | 600.0 | nM | - |
| CHEMBL3728084 | — | IC50 | < | 600.0 | nM | - |
| CHEMBL3732550 | — | IC50 | < | 600.0 | nM | - |
| CHEMBL3729028 | — | IC50 | < | 600.0 | nM | - |
| CHEMBL3729364 | — | IC50 | > | 1200.0 | nM | - |
| CHEMBL3732851 | — | IC50 | < | 600.0 | nM | - |
| CHEMBL3732454 | — | IC50 | < | 600.0 | nM | - |
| CHEMBL3729573 | — | IC50 | < | 600.0 | nM | - |
| CHEMBL3730751 | — | IC50 | < | 600.0 | nM | - |
| CHEMBL3731335 | — | IC50 | < | 600.0 | nM | - |
| CHEMBL3731260 | — | IC50 | < | 600.0 | nM | - |
| CHEMBL3732833 | — | IC50 | < | 600.0 | nM | - |
| CHEMBL3729876 | — | IC50 | < | 600.0 | nM | - |
| CHEMBL3730994 | — | IC50 | < | 600.0 | nM | - |
| CHEMBL3733297 | — | IC50 | < | 600.0 | nM | - |
| CHEMBL3728472 | — | IC50 | < | 600.0 | nM | - |
| CHEMBL3732098 | — | IC50 | < | 600.0 | nM | - |
| CHEMBL3733011 | — | IC50 | < | 600.0 | nM | - |
| CHEMBL3728924 | — | IC50 | < | 600.0 | nM | - |
| CHEMBL3732872 | — | IC50 | < | 600.0 | nM | - |
| CHEMBL3729608 | — | IC50 | < | 600.0 | nM | - |
| CHEMBL3729622 | — | IC50 | < | 600.0 | nM | - |
| CHEMBL3727596 | — | IC50 | > | 1200.0 | nM | - |
| CHEMBL3728373 | — | IC50 | > | 1200.0 | nM | - |