Assay Detail
Binding
CHEMBL3734162
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of PGK1 (unknown origin) pre-incubated with enzyme before 3-phosphoglycerate substrate addition and incubated for 30 mins in presence of NADH and ATP by glyceraldehyde P-dehydrogenase coupling based NADH fluorescence assay
91
Total Activities
91
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Phosphoglycerate kinase inhibitors
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 91 | 6.25 | 9.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3731422 | — | — | 1 | 9.00 |
| CHEMBL3730386 | — | — | 1 | 8.30 |
| CHEMBL3728435 | — | — | 1 | 8.10 |
| CHEMBL1995927 | — | — | 1 | 8.05 |
| CHEMBL3732725 | — | — | 1 | 7.92 |
| CHEMBL3731664 | — | — | 1 | 7.82 |
| CHEMBL3731002 | — | — | 1 | 7.80 |
| CHEMBL3729175 | — | — | 1 | 7.72 |
| CHEMBL3730091 | — | — | 1 | 7.44 |
| CHEMBL3732027 | — | — | 1 | 7.42 |
| CHEMBL3729776 | — | — | 1 | 7.39 |
| CHEMBL3731566 | — | — | 1 | 7.38 |
| CHEMBL3732479 | — | — | 1 | 7.27 |
| CHEMBL3731179 | — | — | 1 | 7.18 |
| CHEMBL3730455 | — | — | 1 | 7.18 |
| CHEMBL3732615 | — | — | 1 | 7.15 |
| CHEMBL3732983 | — | — | 1 | 7.12 |
| CHEMBL3731721 | — | — | 1 | 7.11 |
| CHEMBL3732218 | — | — | 1 | 7.04 |
| CHEMBL3733318 | — | — | 1 | 7.01 |
| CHEMBL3733323 | — | — | 1 | 6.99 |
| CHEMBL3733024 | — | — | 1 | 6.91 |
| CHEMBL3732229 | — | — | 1 | 6.90 |
| CHEMBL3728250 | — | — | 1 | 6.89 |
| CHEMBL3727706 | — | — | 1 | 6.76 |
| CHEMBL3727770 | — | — | 1 | 6.72 |
| CHEMBL3730838 | — | — | 1 | 6.71 |
| CHEMBL3731570 | — | — | 1 | 6.68 |
| CHEMBL3730400 | — | — | 1 | 6.66 |
| CHEMBL3727820 | — | — | 1 | 6.62 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3731422 | — | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL3730386 | — | IC50 | = | 5.0 | nM | 8.30 |
| CHEMBL3728435 | — | IC50 | = | 8.0 | nM | 8.10 |
| CHEMBL1995927 | — | IC50 | = | 9.0 | nM | 8.05 |
| CHEMBL3732725 | — | IC50 | = | 12.0 | nM | 7.92 |
| CHEMBL3731664 | — | IC50 | = | 15.0 | nM | 7.82 |
| CHEMBL3731002 | — | IC50 | = | 16.0 | nM | 7.80 |
| CHEMBL3729175 | — | IC50 | = | 19.0 | nM | 7.72 |
| CHEMBL3730091 | — | IC50 | = | 36.0 | nM | 7.44 |
| CHEMBL3732027 | — | IC50 | = | 38.0 | nM | 7.42 |
| CHEMBL3729776 | — | IC50 | = | 41.0 | nM | 7.39 |
| CHEMBL3731566 | — | IC50 | = | 42.0 | nM | 7.38 |
| CHEMBL3732479 | — | IC50 | = | 54.0 | nM | 7.27 |
| CHEMBL3730455 | — | IC50 | = | 66.0 | nM | 7.18 |
| CHEMBL3731179 | — | IC50 | = | 66.0 | nM | 7.18 |
| CHEMBL3732615 | — | IC50 | = | 71.0 | nM | 7.15 |
| CHEMBL3732983 | — | IC50 | = | 75.0 | nM | 7.12 |
| CHEMBL3731721 | — | IC50 | = | 78.0 | nM | 7.11 |
| CHEMBL3732218 | — | IC50 | = | 91.0 | nM | 7.04 |
| CHEMBL3733318 | — | IC50 | = | 98.0 | nM | 7.01 |
| CHEMBL3733323 | — | IC50 | = | 103.0 | nM | 6.99 |
| CHEMBL3733024 | — | IC50 | = | 122.0 | nM | 6.91 |
| CHEMBL3732229 | — | IC50 | = | 125.0 | nM | 6.90 |
| CHEMBL3728250 | — | IC50 | = | 129.0 | nM | 6.89 |
| CHEMBL3727706 | — | IC50 | = | 173.0 | nM | 6.76 |
| CHEMBL3727770 | — | IC50 | = | 190.0 | nM | 6.72 |
| CHEMBL3730838 | — | IC50 | = | 195.0 | nM | 6.71 |
| CHEMBL3731570 | — | IC50 | = | 210.0 | nM | 6.68 |
| CHEMBL3730400 | — | IC50 | = | 220.0 | nM | 6.66 |
| CHEMBL3727820 | — | IC50 | = | 240.0 | nM | 6.62 |
| CHEMBL3728634 | — | IC50 | = | 252.0 | nM | 6.60 |
| CHEMBL3731180 | — | IC50 | = | 257.0 | nM | 6.59 |
| CHEMBL3729424 | — | IC50 | = | 270.0 | nM | 6.57 |
| CHEMBL3731979 | — | IC50 | = | 320.0 | nM | 6.50 |
| CHEMBL3727853 | — | IC50 | = | 346.0 | nM | 6.46 |
| CHEMBL3730512 | — | IC50 | = | 366.0 | nM | 6.44 |
| CHEMBL3727920 | — | IC50 | = | 385.0 | nM | 6.42 |
| CHEMBL3732267 | — | IC50 | = | 393.0 | nM | 6.41 |
| CHEMBL3731901 | — | IC50 | = | 515.0 | nM | 6.29 |
| CHEMBL3732863 | — | IC50 | = | 550.0 | nM | 6.26 |
| CHEMBL3732931 | — | IC50 | = | 556.0 | nM | 6.25 |
| CHEMBL3728714 | — | IC50 | = | 570.0 | nM | 6.24 |
| CHEMBL3731055 | — | IC50 | = | 596.0 | nM | 6.22 |
| CHEMBL3728173 | — | IC50 | = | 633.0 | nM | 6.20 |
| CHEMBL3733215 | — | IC50 | = | 665.0 | nM | 6.18 |
| CHEMBL3728456 | — | IC50 | = | 710.0 | nM | 6.15 |
| CHEMBL3729640 | — | IC50 | = | 741.0 | nM | 6.13 |
| CHEMBL3728706 | — | IC50 | = | 840.0 | nM | 6.08 |
| CHEMBL3729537 | — | IC50 | = | 884.0 | nM | 6.05 |
| CHEMBL3729183 | — | IC50 | = | 1030.0 | nM | 5.99 |