Assay Detail
Binding
CHEMBL3734284
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Inhibition of GRK3 (unknown origin) after 90 to 120 mins by Kinase-Glo assay
24
Total Activities
24
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
G protein-coupled receptor kinase 3 (CHEMBL1075166) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Hydrazide compounds
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 24 | 6.96 | 8.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3732018 | — | — | 1 | 8.00 |
| CHEMBL3729453 | — | — | 1 | 8.00 |
| CHEMBL3728772 | — | — | 1 | 8.00 |
| CHEMBL3728346 | — | — | 1 | 8.00 |
| CHEMBL3728662 | — | — | 1 | 8.00 |
| CHEMBL3732155 | — | — | 1 | 7.00 |
| CHEMBL3731472 | — | — | 1 | 7.00 |
| CHEMBL3729247 | — | — | 1 | 7.00 |
| CHEMBL3729970 | — | — | 1 | 7.00 |
| CHEMBL3727997 | — | — | 1 | 7.00 |
| CHEMBL3730555 | — | — | 1 | 7.00 |
| CHEMBL3733136 | — | — | 1 | 7.00 |
| CHEMBL3729682 | — | — | 1 | 7.00 |
| CHEMBL3727728 | — | — | 1 | 7.00 |
| CHEMBL3729597 | — | — | 1 | 7.00 |
| CHEMBL3731262 | — | — | 1 | 7.00 |
| CHEMBL3729044 | — | — | 1 | 7.00 |
| CHEMBL3732736 | — | — | 1 | 6.00 |
| CHEMBL3730250 | — | — | 1 | 6.00 |
| CHEMBL3730586 | — | — | 1 | 6.00 |
| CHEMBL3728445 | — | — | 1 | 6.00 |
| CHEMBL3728684 | — | — | 1 | 6.00 |
| CHEMBL3731114 | — | — | 1 | 6.00 |
| CHEMBL3729412 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3732018 | — | Ki | = | 10.0 | nM | 8.00 |
| CHEMBL3729453 | — | Ki | = | 10.0 | nM | 8.00 |
| CHEMBL3728772 | — | Ki | = | 10.0 | nM | 8.00 |
| CHEMBL3728346 | — | Ki | = | 10.0 | nM | 8.00 |
| CHEMBL3728662 | — | Ki | = | 10.0 | nM | 8.00 |
| CHEMBL3732155 | — | Ki | = | 100.0 | nM | 7.00 |
| CHEMBL3731472 | — | Ki | = | 100.0 | nM | 7.00 |
| CHEMBL3729247 | — | Ki | = | 100.0 | nM | 7.00 |
| CHEMBL3729970 | — | Ki | = | 100.0 | nM | 7.00 |
| CHEMBL3727997 | — | Ki | = | 100.0 | nM | 7.00 |
| CHEMBL3730555 | — | Ki | = | 100.0 | nM | 7.00 |
| CHEMBL3733136 | — | Ki | = | 100.0 | nM | 7.00 |
| CHEMBL3729682 | — | Ki | = | 100.0 | nM | 7.00 |
| CHEMBL3727728 | — | Ki | = | 100.0 | nM | 7.00 |
| CHEMBL3729597 | — | Ki | = | 100.0 | nM | 7.00 |
| CHEMBL3731262 | — | Ki | = | 100.0 | nM | 7.00 |
| CHEMBL3729044 | — | Ki | = | 100.0 | nM | 7.00 |
| CHEMBL3732736 | — | Ki | = | 1000.0 | nM | 6.00 |
| CHEMBL3730250 | — | Ki | = | 1000.0 | nM | 6.00 |
| CHEMBL3730586 | — | Ki | = | 1000.0 | nM | 6.00 |
| CHEMBL3728445 | — | Ki | = | 1000.0 | nM | 6.00 |
| CHEMBL3728684 | — | Ki | = | 1000.0 | nM | 6.00 |
| CHEMBL3731114 | — | Ki | = | 1000.0 | nM | 6.00 |
| CHEMBL3729412 | — | Ki | > | 10000.0 | nM | - |