Assay Detail
Binding
CHEMBL3734546
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of STIM1/Orai1 in rat RBL2H3 cells assessed as inhibition of upslope incubated for 5 mins followed by thapsigargin addition for 25 mins measured for 7 secs by fluo4-AM dye-based FLIPR assay
84
Total Activities
84
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Rattus norvegicus |
| Cell Type | RBL-2H3 |
| Confidence | 7 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Compounds that modulate intracellular calcium
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 84 | 6.22 | 6.22 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3732761 | — | — | 1 | 6.22 |
| CHEMBL3728969 | — | — | 1 | 6.22 |
| CHEMBL3729739 | — | — | 1 | 6.22 |
| CHEMBL3732450 | — | — | 1 | 6.22 |
| CHEMBL3727649 | — | — | 1 | 6.22 |
| CHEMBL3731310 | — | — | 1 | 6.22 |
| CHEMBL3731030 | — | — | 1 | 6.22 |
| CHEMBL3733059 | — | — | 1 | 6.22 |
| CHEMBL3731485 | — | — | 1 | 6.22 |
| CHEMBL3727447 | — | — | 1 | 6.22 |
| CHEMBL3733237 | — | — | 1 | 6.22 |
| CHEMBL3727600 | — | — | 1 | 6.22 |
| CHEMBL3731964 | — | — | 1 | 6.22 |
| CHEMBL3728704 | — | — | 1 | - |
| CHEMBL3729771 | — | — | 1 | - |
| CHEMBL3731651 | — | — | 1 | - |
| CHEMBL3729158 | — | — | 1 | - |
| CHEMBL3730254 | — | — | 1 | - |
| CHEMBL3732677 | — | — | 1 | - |
| CHEMBL3728713 | — | — | 1 | - |
| CHEMBL3729234 | — | — | 1 | - |
| CHEMBL3728323 | — | — | 1 | - |
| CHEMBL3728931 | — | — | 1 | - |
| CHEMBL3733040 | — | — | 1 | - |
| CHEMBL3730009 | — | — | 1 | - |
| CHEMBL3732779 | — | — | 1 | - |
| CHEMBL3727734 | — | — | 1 | - |
| CHEMBL3732110 | — | — | 1 | - |
| CHEMBL3731765 | — | — | 1 | - |
| CHEMBL3730176 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3732761 | — | IC50 | = | 600.0 | nM | 6.22 |
| CHEMBL3728969 | — | IC50 | = | 600.0 | nM | 6.22 |
| CHEMBL3729739 | — | IC50 | = | 600.0 | nM | 6.22 |
| CHEMBL3732450 | — | IC50 | = | 600.0 | nM | 6.22 |
| CHEMBL3727649 | — | IC50 | = | 600.0 | nM | 6.22 |
| CHEMBL3731310 | — | IC50 | = | 600.0 | nM | 6.22 |
| CHEMBL3731030 | — | IC50 | = | 600.0 | nM | 6.22 |
| CHEMBL3733059 | — | IC50 | = | 600.0 | nM | 6.22 |
| CHEMBL3731485 | — | IC50 | = | 600.0 | nM | 6.22 |
| CHEMBL3727447 | — | IC50 | = | 600.0 | nM | 6.22 |
| CHEMBL3733237 | — | IC50 | = | 600.0 | nM | 6.22 |
| CHEMBL3727600 | — | IC50 | = | 600.0 | nM | 6.22 |
| CHEMBL3731964 | — | IC50 | = | 600.0 | nM | 6.22 |
| CHEMBL3729841 | — | IC50 | < | 600.0 | nM | - |
| CHEMBL3727872 | — | IC50 | - | — | - | |
| CHEMBL3728875 | — | IC50 | < | 600.0 | nM | - |
| CHEMBL3727938 | — | IC50 | < | 600.0 | nM | - |
| CHEMBL3732114 | — | IC50 | < | 600.0 | nM | - |
| CHEMBL3729900 | — | IC50 | < | 600.0 | nM | - |
| CHEMBL3729109 | — | IC50 | < | 600.0 | nM | - |
| CHEMBL3730610 | — | IC50 | - | — | - | |
| CHEMBL3729551 | — | IC50 | < | 600.0 | nM | - |
| CHEMBL3733355 | — | IC50 | < | 600.0 | nM | - |
| CHEMBL3727989 | — | IC50 | < | 600.0 | nM | - |
| CHEMBL3728468 | — | IC50 | - | — | - | |
| CHEMBL3727611 | — | IC50 | - | — | - | |
| CHEMBL3731488 | — | IC50 | < | 600.0 | nM | - |
| CHEMBL3728218 | — | IC50 | - | — | - | |
| CHEMBL3732620 | — | IC50 | < | 600.0 | nM | - |
| CHEMBL3728855 | — | IC50 | < | 600.0 | nM | - |
| CHEMBL3732547 | — | IC50 | < | 600.0 | nM | - |
| CHEMBL3729234 | — | IC50 | - | — | - | |
| CHEMBL3730176 | — | IC50 | - | — | - | |
| CHEMBL3731765 | — | IC50 | < | 600.0 | nM | - |
| CHEMBL3732110 | — | IC50 | - | — | - | |
| CHEMBL3727734 | — | IC50 | < | 600.0 | nM | - |
| CHEMBL3732779 | — | IC50 | < | 600.0 | nM | - |
| CHEMBL3730009 | — | IC50 | < | 600.0 | nM | - |
| CHEMBL3733040 | — | IC50 | < | 600.0 | nM | - |
| CHEMBL3728931 | — | IC50 | > | 1200.0 | nM | - |
| CHEMBL3728323 | — | IC50 | < | 600.0 | nM | - |
| CHEMBL3729101 | — | IC50 | < | 600.0 | nM | - |
| CHEMBL3728713 | — | IC50 | - | — | - | |
| CHEMBL3732677 | — | IC50 | < | 600.0 | nM | - |
| CHEMBL3730254 | — | IC50 | < | 600.0 | nM | - |
| CHEMBL3729158 | — | IC50 | < | 600.0 | nM | - |
| CHEMBL3731651 | — | IC50 | < | 600.0 | nM | - |
| CHEMBL3729771 | — | IC50 | < | 600.0 | nM | - |
| CHEMBL3728704 | — | IC50 | < | 600.0 | nM | - |
| CHEMBL3730740 | — | IC50 | < | 600.0 | nM | - |