Assay Detail
Functional
CHEMBL3734548
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Antagonist activity at MrgX1 (unknown origin) by beta-lactamase reporter gene assay
16
Total Activities
16
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Mas-related G-protein coupled receptor member X1 (CHEMBL5850) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Methods and compositions for treating or preventing pruritis
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 16 | 6.76 | 7.30 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3343995 | — | — | 1 | 7.30 |
| CHEMBL3727438 | — | — | 1 | 7.19 |
| CHEMBL3730717 | — | — | 1 | 7.10 |
| CHEMBL3730500 | — | — | 1 | 7.05 |
| CHEMBL3730405 | — | — | 1 | 6.91 |
| CHEMBL3730599 | — | — | 1 | 6.85 |
| CHEMBL3731811 | — | — | 1 | 6.79 |
| CHEMBL3727861 | — | — | 1 | 6.78 |
| CHEMBL3730179 | — | — | 1 | 6.70 |
| CHEMBL3729794 | — | — | 1 | 6.68 |
| CHEMBL3728505 | — | — | 1 | 6.61 |
| CHEMBL3731844 | — | — | 1 | 6.60 |
| CHEMBL3732603 | — | — | 1 | 6.54 |
| CHEMBL3733177 | — | — | 1 | 6.43 |
| CHEMBL3728009 | — | — | 1 | 6.38 |
| CHEMBL145103 | — | — | 1 | 6.25 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3343995 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3727438 | — | IC50 | = | 64.0 | nM | 7.19 |
| CHEMBL3730717 | — | IC50 | = | 80.0 | nM | 7.10 |
| CHEMBL3730500 | — | IC50 | = | 90.0 | nM | 7.05 |
| CHEMBL3730405 | — | IC50 | = | 124.0 | nM | 6.91 |
| CHEMBL3730599 | — | IC50 | = | 140.0 | nM | 6.85 |
| CHEMBL3731811 | — | IC50 | = | 163.0 | nM | 6.79 |
| CHEMBL3727861 | — | IC50 | = | 165.0 | nM | 6.78 |
| CHEMBL3730179 | — | IC50 | = | 200.0 | nM | 6.70 |
| CHEMBL3729794 | — | IC50 | = | 209.0 | nM | 6.68 |
| CHEMBL3728505 | — | IC50 | = | 244.0 | nM | 6.61 |
| CHEMBL3731844 | — | IC50 | = | 252.0 | nM | 6.60 |
| CHEMBL3732603 | — | IC50 | = | 290.0 | nM | 6.54 |
| CHEMBL3733177 | — | IC50 | = | 375.0 | nM | 6.43 |
| CHEMBL3728009 | — | IC50 | = | 418.0 | nM | 6.38 |
| CHEMBL145103 | — | IC50 | = | 556.0 | nM | 6.25 |