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Assay Detail

CHEMBL3742625

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Physicochemical
Antioxidant activity assessed as galvinoxyl radical scavenging activity measured over 30 mins by spectrophotometry
7
Total Activities
7
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Physicochemical
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Publication

Exploring cinnamic acid scaffold: development of promising neuroprotective lipophilic antioxidants
Chavarria D, Silva T, Martins D, Bravo J, Summavielle T, Garrido J, Borges F
Medchemcomm (2015) 6 : 1043 -1053
· DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 7 5.11 5.60

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL507378 DEMETHYLENATED PIPERIC ACID 1 5.60
CHEMBL153 TROLOX 1 5.47
CHEMBL3742265 1 5.32
CHEMBL32749 FERULATE -1.0 1 4.58
CHEMBL145 CAFFEIC ACID 3.0 1 4.57
CHEMBL320295 O,O'-DIMETHYLCAFFEIC ACID 1 -
CHEMBL3741423 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL507378 DEMETHYLENATED PIPERIC ACID IC50 = 2500.0 nM 5.60
CHEMBL153 TROLOX IC50 = 3400.0 nM 5.47
CHEMBL3742265 IC50 = 4800.0 nM 5.32
CHEMBL32749 FERULATE IC50 = 26500.0 nM 4.58
CHEMBL145 CAFFEIC ACID IC50 = 27000.0 nM 4.57
CHEMBL320295 O,O'-DIMETHYLCAFFEIC ACID IC50 - -
CHEMBL3741423 IC50 - -