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Assay Detail

CHEMBL3742981

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antibiofilm activity against Pseudoalteromonas lipolytica TC8 assessed as reduction in adhesion after 15 hrs by Syto61 based-fluorescence analysis relative to control
8
Total Activities
8
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Pseudoalteromonas lipolytica
Confidence 1 — Organism
Curated By Autocuration

Target

Pseudoalteromonas lipolytica (CHEMBL4296594)
Type ORGANISM
Organism Pseudoalteromonas lipolytica

Publication

Click-based synthesis of bromotyrosine alkaloid analogs as potential anti-biofilm leads for SAR studies.
Andjouh S, Blache Y.
Bioorg Med Chem Lett (2015) 25 : 5762 -5766
PubMed 26564265 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 8 4.31 4.75

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL174 AMPICILLIN 4.0 1 4.75
CHEMBL3739616 1 4.17
CHEMBL3739688 1 4.02
CHEMBL3741233 1 -
CHEMBL3739976 1 -
CHEMBL3742346 1 -
CHEMBL3739635 1 -
CHEMBL3741894 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL174 AMPICILLIN EC50 = 17900.0 nM 4.75
CHEMBL3739616 EC50 = 67800.0 nM 4.17
CHEMBL3739688 EC50 = 96000.0 nM 4.02
CHEMBL3741233 EC50 = 123600.0 nM -
CHEMBL3739976 EC50 = 170500.0 nM -
CHEMBL3742346 EC50 = 113200.0 nM -
CHEMBL3739635 EC50 = 104400.0 nM -
CHEMBL3741894 EC50 = 134200.0 nM -