Assay Detail
Binding
CHEMBL3748085
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Antiviral activity against HIV1 assessed as inhibition of integrase
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Human immunodeficiency virus 1 |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Human immunodeficiency virus type 1 integrase (CHEMBL3471) ↗| Type | SINGLE PROTEIN |
| Organism | Human immunodeficiency virus 1 |
Publication
New Frontiers in Druggability.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 2 | 7.16 | 7.16 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3747158 | — | — | 1 | 7.16 |
| CHEMBL1230654 | — | — | 1 | 7.16 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3747158 | — | EC50 | = | 69.0 | nM | 7.16 |
| CHEMBL1230654 | — | EC50 | = | 69.0 | nM | 7.16 |