Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL3750554

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of Staphylococcus aureus mtgA after 30 mins by continous fluorescence assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Staphylococcus aureus
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

Unchecked (CHEMBL612545)
Type UNCHECKED

Publication

Structure-Activity Relationships of Novel Tryptamine-Based Inhibitors of Bacterial Transglycosylase.
Sosič I, Anderluh M, Sova M, Gobec M, Mlinarič Raščan I, Derouaux A, Amoroso A, Terrak M, Breukink E, Gobec S.
J Med Chem (2015) 58 : 9712 -9721
PubMed 26588190 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 4.57 4.57

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL3746902 1 4.57

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL3746902 IC50 = 27000.0 nM 4.57