Assay Detail
Binding
CHEMBL3755504
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Antagonist activity at TRPV1 (unknown origin) in DRG neurons
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Transient receptor potential cation channel subfamily V member 1 (CHEMBL4794) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
TRPA1 channels as targets for resveratrol and related stilbenoids.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 4.52 | 4.52 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL186366 | PINOSYLVIN METHYL ETHER | — | 1 | 4.52 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL186366 | PINOSYLVIN METHYL ETHER | IC50 | = | 30000.0 | nM | 4.52 |