Assay Detail
Functional
CHEMBL3756443
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of serum-opsonized zymosan-induced oxidative burst in whole blood (unknown origin)
9
Total Activities
9
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Not specified |
| Tissue | Blood |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Oxidative burst inhibition, cytotoxicity and antibacterial acriquinoline alkaloids from Citrus reticulate (Blanco).
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 9 | 4.92 | 5.35 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3754791 | — | — | 1 | 5.35 |
| CHEMBL140796 | ISOPIMPINELLIN | — | 1 | 5.03 |
| CHEMBL465808 | ATALANTOFLAVONE | — | 1 | 4.98 |
| CHEMBL521 | IBUPROFEN | 4.0 | 1 | 4.95 |
| CHEMBL325864 | SCOPARONE | — | 1 | 4.94 |
| CHEMBL3753940 | — | — | 1 | 4.79 |
| CHEMBL3752565 | — | — | 1 | 4.76 |
| CHEMBL1928409 | SUBEROSIN | — | 1 | 4.74 |
| CHEMBL3752540 | — | — | 1 | 4.70 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3754791 | — | IC50 | = | 4500.0 | nM | 5.35 |
| CHEMBL140796 | ISOPIMPINELLIN | IC50 | = | 9400.0 | nM | 5.03 |
| CHEMBL465808 | ATALANTOFLAVONE | IC50 | = | 10500.0 | nM | 4.98 |
| CHEMBL521 | IBUPROFEN | IC50 | = | 11200.0 | nM | 4.95 |
| CHEMBL325864 | SCOPARONE | IC50 | = | 11400.0 | nM | 4.94 |
| CHEMBL3753940 | — | IC50 | = | 16400.0 | nM | 4.79 |
| CHEMBL3752565 | — | IC50 | = | 17200.0 | nM | 4.76 |
| CHEMBL1928409 | SUBEROSIN | IC50 | = | 18300.0 | nM | 4.74 |
| CHEMBL3752540 | — | IC50 | = | 20100.0 | nM | 4.70 |