Assay Detail
Binding
CHEMBL3766474
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Binding affinity to carbonic anhydrase2 (unknown origin) by surface plasmon resonance assay
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Novel Small Molecule Inhibitors of Choline Kinase Identified by Fragment-Based Drug Discovery.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Kd | 3 | 3.11 | 3.31 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3763993 | — | — | 1 | 3.31 |
| CHEMBL3764475 | — | — | 1 | 3.17 |
| CHEMBL3763196 | — | — | 1 | 2.85 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3763993 | — | Kd | = | 490000.0 | nM | 3.31 |
| CHEMBL3764475 | — | Kd | = | 670000.0 | nM | 3.17 |
| CHEMBL3763196 | — | Kd | = | 1400000.0 | nM | 2.85 |