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Assay Detail

CHEMBL3767658

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Binding affinity to vasopressin 1a receptor (unknown origin)
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Vasopressin V1a receptor (CHEMBL1889)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Flexible analogues of WAY-267,464: Synthesis and pharmacology at the human oxytocin and vasopressin 1a receptors.
Jorgensen WT, Gulliver DW, Werry EL, Reekie T, Connor M, Kassiou M.
Eur J Med Chem (2016) 108 : 730 -740
PubMed 26741855 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 1 6.95 6.95

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL3763342 1 6.95

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL3763342 Ki = 113.0 nM 6.95