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Assay Detail

CHEMBL3768093

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Binding
Binding affinity to wild type Magnetospirillum gryphiswaldense cereblon isoform 4 by FRET assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Magnetospirillum gryphiswaldense
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Cereblon isoform 4 (CHEMBL3763007)
Type SINGLE PROTEIN
Organism Magnetospirillum gryphiswaldense

Publication

A FRET-Based Assay for the Identification and Characterization of Cereblon Ligands.
Boichenko I, Deiss S, Bär K, Hartmann MD, Hernandez Alvarez B.
J Med Chem (2016) 59 : 770 -774
PubMed 26730808 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Kd 1 5.48 5.48

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL3764647 1 5.48

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL3764647 Kd = 3300.0 nM 5.48