Assay Detail
Binding
CHEMBL3771489
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Inhibition of BRPF1B (unknown origin) by Alpha Screen assay
25
Total Activities
25
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Discovery of a Chemical Tool Inhibitor Targeting the Bromodomains of TRIM24 and BRPF.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 25 | 6.19 | 6.57 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3770173 | — | — | 1 | 6.57 |
| CHEMBL3770004 | — | — | 1 | 6.57 |
| CHEMBL3770971 | — | — | 1 | 6.57 |
| CHEMBL3771151 | — | — | 1 | 6.54 |
| CHEMBL3769887 | — | — | 1 | 6.54 |
| CHEMBL3771106 | — | — | 1 | 6.51 |
| CHEMBL1346130 | — | — | 1 | 6.48 |
| CHEMBL3769965 | — | — | 1 | 6.47 |
| CHEMBL3771002 | — | — | 1 | 6.47 |
| CHEMBL3770886 | — | — | 1 | 6.38 |
| CHEMBL3770391 | — | — | 1 | 6.37 |
| CHEMBL3770465 | — | — | 1 | 6.37 |
| CHEMBL3771226 | — | — | 1 | 6.29 |
| CHEMBL3770652 | — | — | 1 | 6.23 |
| CHEMBL3770456 | — | — | 1 | 6.18 |
| CHEMBL3770259 | — | — | 1 | 6.18 |
| CHEMBL3771005 | — | — | 1 | 6.17 |
| CHEMBL3770048 | — | — | 1 | 6.10 |
| CHEMBL3770861 | — | — | 1 | 5.98 |
| CHEMBL3771154 | — | — | 1 | 5.93 |
| CHEMBL3771239 | — | — | 1 | 5.85 |
| CHEMBL3770384 | — | — | 1 | 5.65 |
| CHEMBL3771230 | — | — | 1 | 5.57 |
| CHEMBL3770810 | — | — | 1 | 5.51 |
| CHEMBL3769732 | — | — | 1 | 5.17 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3770173 | — | IC50 | = | 270.0 | nM | 6.57 |
| CHEMBL3770004 | — | IC50 | = | 270.0 | nM | 6.57 |
| CHEMBL3770971 | — | IC50 | = | 270.0 | nM | 6.57 |
| CHEMBL3771151 | — | IC50 | = | 290.0 | nM | 6.54 |
| CHEMBL3769887 | — | IC50 | = | 290.0 | nM | 6.54 |
| CHEMBL3771106 | — | IC50 | = | 310.0 | nM | 6.51 |
| CHEMBL1346130 | — | IC50 | = | 330.0 | nM | 6.48 |
| CHEMBL3769965 | — | IC50 | = | 340.0 | nM | 6.47 |
| CHEMBL3771002 | — | IC50 | = | 340.0 | nM | 6.47 |
| CHEMBL3770886 | — | IC50 | = | 420.0 | nM | 6.38 |
| CHEMBL3770391 | — | IC50 | = | 430.0 | nM | 6.37 |
| CHEMBL3770465 | — | IC50 | = | 430.0 | nM | 6.37 |
| CHEMBL3771226 | — | IC50 | = | 510.0 | nM | 6.29 |
| CHEMBL3770652 | — | IC50 | = | 590.0 | nM | 6.23 |
| CHEMBL3770456 | — | IC50 | = | 660.0 | nM | 6.18 |
| CHEMBL3770259 | — | IC50 | = | 660.0 | nM | 6.18 |
| CHEMBL3771005 | — | IC50 | = | 680.0 | nM | 6.17 |
| CHEMBL3770048 | — | IC50 | = | 790.0 | nM | 6.10 |
| CHEMBL3770861 | — | IC50 | = | 1050.0 | nM | 5.98 |
| CHEMBL3771154 | — | IC50 | = | 1170.0 | nM | 5.93 |
| CHEMBL3771239 | — | IC50 | = | 1400.0 | nM | 5.85 |
| CHEMBL3770384 | — | IC50 | = | 2240.0 | nM | 5.65 |
| CHEMBL3771230 | — | IC50 | = | 2680.0 | nM | 5.57 |
| CHEMBL3770810 | — | IC50 | = | 3100.0 | nM | 5.51 |
| CHEMBL3769732 | — | IC50 | = | 6720.0 | nM | 5.17 |