Assay Detail
Binding
CHEMBL3773446
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Inhibition of BRD9 (unknown origin) incubated in dark for 30 mins by TR-FRET assay
14
Total Activities
14
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Discovery of I-BRD9, a Selective Cell Active Chemical Probe for Bromodomain Containing Protein 9 Inhibition.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 14 | 7.05 | 8.10 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3770188 | — | — | 1 | 8.10 |
| CHEMBL3769944 | — | — | 1 | 8.00 |
| CHEMBL3769688 | — | — | 1 | 7.90 |
| CHEMBL3769855 | — | — | 1 | 7.90 |
| CHEMBL3770949 | — | — | 1 | 7.80 |
| CHEMBL3769509 | — | — | 1 | 7.40 |
| CHEMBL3769628 | — | — | 1 | 7.40 |
| CHEMBL3769507 | — | — | 1 | 7.30 |
| CHEMBL3770367 | — | — | 1 | 7.10 |
| CHEMBL3770039 | — | — | 1 | 6.90 |
| CHEMBL3769979 | — | — | 1 | 6.70 |
| CHEMBL3770716 | — | — | 1 | 5.50 |
| CHEMBL3771218 | — | — | 1 | 5.40 |
| CHEMBL3771308 | — | — | 1 | 5.30 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3770188 | — | IC50 | = | 7.943 | nM | 8.10 |
| CHEMBL3769944 | — | IC50 | = | 10.0 | nM | 8.00 |
| CHEMBL3769688 | — | IC50 | = | 12.59 | nM | 7.90 |
| CHEMBL3769855 | — | IC50 | = | 12.59 | nM | 7.90 |
| CHEMBL3770949 | — | IC50 | = | 15.85 | nM | 7.80 |
| CHEMBL3769509 | — | IC50 | = | 39.81 | nM | 7.40 |
| CHEMBL3769628 | — | IC50 | = | 39.81 | nM | 7.40 |
| CHEMBL3769507 | — | IC50 | = | 50.12 | nM | 7.30 |
| CHEMBL3770367 | — | IC50 | = | 79.43 | nM | 7.10 |
| CHEMBL3770039 | — | IC50 | = | 125.89 | nM | 6.90 |
| CHEMBL3769979 | — | IC50 | = | 199.53 | nM | 6.70 |
| CHEMBL3770716 | — | IC50 | = | 3162.28 | nM | 5.50 |
| CHEMBL3771218 | — | IC50 | = | 3981.07 | nM | 5.40 |
| CHEMBL3771308 | — | IC50 | = | 5011.87 | nM | 5.30 |