Assay Detail
Binding
CHEMBL3777314
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Binding affinity to angiotensin II receptor (unknown origin)
5
Total Activities
5
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Tactical Approaches to Interconverting GPCR Agonists and Antagonists.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 5 | 8.53 | 9.15 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL217673 | — | — | 1 | 9.15 |
| CHEMBL39959 | — | — | 1 | 8.82 |
| CHEMBL289614 | — | — | 1 | 8.68 |
| CHEMBL3394209 | — | — | 1 | 8.09 |
| CHEMBL3394207 | — | — | 1 | 7.91 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL217673 | — | Ki | = | 0.7 | nM | 9.15 |
| CHEMBL39959 | — | Ki | = | 1.5 | nM | 8.82 |
| CHEMBL289614 | — | Ki | = | 2.1 | nM | 8.68 |
| CHEMBL3394209 | — | Ki | = | 8.2 | nM | 8.09 |
| CHEMBL3394207 | — | Ki | = | 12.3 | nM | 7.91 |