Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL3782199

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antioxidant activity in human HepG2 cells assessed as decrease in fluorescence level after 2.5 hrs measured every 5 mins for 1 hr by DCFH-DA staining based fluorescence assay
4
Total Activities
3
Compounds Tested
2
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type HepG2
Confidence 1 — Organism
Curated By Autocuration

Target

HepG2 (CHEMBL395)
Type CELL-LINE
Organism Homo sapiens

Publication

Protective effects of kaempferol against reactive oxygen species-induced hemolysis and its antiproliferative activity on human cancer cells.
Liao W, Chen L, Ma X, Jiao R, Li X, Wang Y.
Eur J Med Chem (2016) 114 : 24 -32
PubMed 26974372 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 3 5.18 5.33
Activity 1 - -

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL50 QUERCETIN 3.0 1 5.33
CHEMBL150 KAEMPFEROL 1.0 2 5.11
CHEMBL90568 DIOSMETIN 1 5.10

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL50 QUERCETIN EC50 = 4630.0 nM 5.33
CHEMBL150 KAEMPFEROL EC50 = 7740.0 nM 5.11
CHEMBL90568 DIOSMETIN EC50 = 7980.0 nM 5.10
CHEMBL150 KAEMPFEROL Activity - -