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Assay Detail

CHEMBL3782489

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiviral activity against Human coxsackievirus B2 infected in african green monkey Vero cells after 24 to 36 hrs by MTS-based CPE reduction assay
5
Total Activities
5
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Coxsackievirus B2
Cell Type Vero
Confidence 1 — Organism
Curated By Autocuration

Target

Coxsackievirus B2 (CHEMBL613202)
Type ORGANISM
Organism Coxsackievirus B2

Publication

Identification and Structure-Activity Relationships of Diarylhydrazides as Novel Potent and Selective Human Enterovirus Inhibitors.
Han X, Sun N, Wu H, Guo D, Tien P, Dong C, Wu S, Zhou HB.
J Med Chem (2016) 59 : 2139 -2150
PubMed 26885567 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 5 7.95 9.30

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL3779938 1 9.30
CHEMBL3781846 1 9.05
CHEMBL3780944 1 8.80
CHEMBL283403 ENVIROXIME 2.0 1 6.82
CHEMBL3781624 1 5.80

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL3779938 EC50 = 0.5 nM 9.30
CHEMBL3781846 EC50 = 0.9 nM 9.05
CHEMBL3780944 EC50 = 1.6 nM 8.80
CHEMBL283403 ENVIROXIME EC50 = 150.0 nM 6.82
CHEMBL3781624 EC50 = 1570.0 nM 5.80