Assay Detail
Binding
CHEMBL3784259
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Binding affinity to carbonic anhydrase-2 (unknown origin)
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
On the enthalpic preference of fragment binding
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Kd | 2 | 6.83 | 7.57 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL302715 | — | — | 1 | 7.57 |
| CHEMBL27601 | BENZENESULFONAMIDE | — | 1 | 6.08 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL302715 | — | Kd | = | 27.0 | nM | 7.57 |
| CHEMBL27601 | BENZENESULFONAMIDE | Kd | = | 839.0 | nM | 6.08 |