Assay Detail
Binding
CHEMBL3784756
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of PI3Kdelta (unknown origin)
10
Total Activities
10
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform (CHEMBL3130) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Potent, Selective, and Orally Bioavailable Inhibitors of VPS34 Provide Chemical Tools to Modulate Autophagy in Vivo.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 10 | 5.67 | 6.30 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3780339 | — | — | 1 | 6.30 |
| CHEMBL3781926 | — | — | 1 | 6.13 |
| CHEMBL3781466 | — | — | 1 | 6.09 |
| CHEMBL3781415 | — | — | 1 | 5.92 |
| CHEMBL3780029 | — | — | 1 | 5.54 |
| CHEMBL3781615 | — | — | 1 | 5.43 |
| CHEMBL3780762 | — | — | 1 | 5.38 |
| CHEMBL3781916 | — | — | 1 | 5.16 |
| CHEMBL3781634 | — | — | 1 | 5.07 |
| CHEMBL3781020 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3780339 | — | IC50 | = | 500.0 | nM | 6.30 |
| CHEMBL3781926 | — | IC50 | = | 740.0 | nM | 6.13 |
| CHEMBL3781466 | — | IC50 | = | 820.0 | nM | 6.09 |
| CHEMBL3781415 | — | IC50 | = | 1200.0 | nM | 5.92 |
| CHEMBL3780029 | — | IC50 | = | 2900.0 | nM | 5.54 |
| CHEMBL3781615 | — | IC50 | = | 3700.0 | nM | 5.43 |
| CHEMBL3780762 | — | IC50 | = | 4200.0 | nM | 5.38 |
| CHEMBL3781916 | — | IC50 | = | 7000.0 | nM | 5.16 |
| CHEMBL3781634 | — | IC50 | = | 8500.0 | nM | 5.07 |
| CHEMBL3781020 | — | IC50 | > | 9100.0 | nM | - |