Assay Detail
Binding
CHEMBL3796289
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of recombinant human CK2 holoenzyme using RRRADDSDDDDD as substrate measured after 10 mins at 37 degC by radiometric kinase assay in presence of [gamma-32P]ATP
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 5 — Multiple protein complex / RNA |
| Curated By | Autocuration |
Publication
Design and synthesis of novel protein kinase CK2 inhibitors on the base of 4-aminothieno[2,3-d]pyrimidines.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 1 | 7.22 | 7.22 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL29898 | QUINALIZARIN | — | 1 | 7.22 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL29898 | QUINALIZARIN | Ki | = | 60.0 | nM | 7.22 |