Assay Detail
Binding
CHEMBL3807747
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of HIV1 NL4-3 Env-induced cell-cell fusion between viral envelope expressing African green monkey COS cells to CXCR4 receptor expressing human TZM-bl cells after overnight incubation by Bright-Glo luciferase assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Human immunodeficiency virus 1 |
| Cell Type | COS |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Aloperine and Its Derivatives as a New Class of HIV-1 Entry Inhibitors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 1 | 5.92 | 5.92 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3329704 | — | — | 1 | 5.92 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3329704 | — | EC50 | = | 1200.0 | nM | 5.92 |