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Assay Detail

CHEMBL3812646

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Functional
Antiviral activity against HCV genotype 3a NC009824 assessed as decrease in HCV replicon RNA replication by taqman assay based cell based replicon method
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Hepacivirus hominis
Confidence 1 — Organism
Curated By Autocuration

Target

Hepatitis C virus (CHEMBL379)
Type ORGANISM
Organism Hepacivirus hominis

Publication

Discovery of fused tricyclic core containing HCV NS5A inhibitors with pan-genotype activity.
Yu W, Coburn CA, Yang DY, Meinke PT, Wong M, Rosenblum SB, Chen KX, Njoroge GF, Chen L, Dwyer MP, Jiang Y, Nair AG, Selyutin O, Tong L, Zeng Q, Zhong B, Ji T, Hu B, Agrawal S, Xia E, Zhai Y, Liu R, Kong R, Ingravallo P, Asante-Appiah E, Nomeir A, Fells J, Kozlowski JA.
Bioorg Med Chem Lett (2016) 26 : 3158 -3162
PubMed 27180013 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 1 10.70 10.70

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL3039514 ELBASVIR 4.0 1 10.70

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL3039514 ELBASVIR EC50 = 0.02 nM 10.70