Assay Detail
Binding
CHEMBL3812915
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Displacement of [3H]CP 55940 from human CB1 receptor after 1 hr by liquid scintillation spectrometry
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Discovery of KLS-13019, a Cannabidiol-Derived Neuroprotective Agent, with Improved Potency, Safety, and Permeability.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 7.72 | 7.96 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3809355 | — | — | 1 | 7.96 |
| CHEMBL125061 | — | — | 1 | 7.48 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3809355 | — | Ki | = | 11.0 | nM | 7.96 |
| CHEMBL125061 | — | Ki | = | 33.0 | nM | 7.48 |