Assay Detail
Binding
CHEMBL3820060
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Binding affinity to human dopamine D4 receptor by radioligand displacement assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Development of CNS multi-receptor ligands: Modification of known D2 pharmacophores.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 1 | 10.18 | 10.18 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL297302 | BENPERIDOL | 3.0 | 1 | 10.18 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL297302 | BENPERIDOL | Ki | = | 0.066 | nM | 10.18 |