Assay Detail
Binding
CHEMBL3824477
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Agonist activity at human GLP1R expressed in HEK293 cells after 5 hrs by luciferase reporter gene assay
85
Total Activities
85
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Cell Type | HEK293 |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Synthesis and Pharmacological Characterization of Novel Glucagon-like Peptide-2 (GLP-2) Analogues with Low Systemic Clearance.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 85 | 7.25 | 8.06 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4299664 | — | — | 1 | 8.06 |
| CHEMBL3822701 | — | — | 1 | 8.05 |
| CHEMBL4299677 | — | — | 1 | 8.00 |
| CHEMBL3822593 | — | — | 1 | 7.80 |
| CHEMBL4299655 | — | — | 1 | 7.68 |
| CHEMBL3823755 | — | — | 1 | 7.50 |
| CHEMBL3822625 | — | — | 1 | 7.41 |
| CHEMBL3824159 | — | — | 1 | 7.40 |
| CHEMBL3823411 | — | — | 1 | 7.35 |
| CHEMBL3822981 | — | — | 1 | 7.25 |
| CHEMBL3823448 | — | — | 1 | 7.22 |
| CHEMBL3823334 | — | — | 1 | 7.16 |
| CHEMBL3823889 | — | — | 1 | 7.10 |
| CHEMBL3823221 | — | — | 1 | 7.08 |
| CHEMBL3823421 | — | — | 1 | 7.05 |
| CHEMBL3822975 | — | — | 1 | 7.00 |
| CHEMBL3823878 | — | — | 1 | 6.96 |
| CHEMBL3823876 | — | — | 1 | 6.92 |
| CHEMBL3823835 | — | — | 1 | 6.89 |
| CHEMBL3823333 | — | — | 1 | 6.75 |
| CHEMBL3823760 | — | — | 1 | 6.52 |
| CHEMBL2177395 | — | — | 1 | 6.28 |
| CHEMBL3822636 | — | — | 1 | - |
| CHEMBL4299631 | — | — | 1 | - |
| CHEMBL3822928 | — | — | 1 | - |
| CHEMBL3824278 | — | — | 1 | - |
| CHEMBL3823643 | — | — | 1 | - |
| CHEMBL4299662 | — | — | 1 | - |
| CHEMBL3822459 | — | — | 1 | - |
| CHEMBL3823976 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4299664 | — | EC50 | = | 8.8 | nM | 8.06 |
| CHEMBL3822701 | — | EC50 | = | 8.9 | nM | 8.05 |
| CHEMBL4299677 | — | EC50 | = | 10.0 | nM | 8.00 |
| CHEMBL3822593 | — | EC50 | = | 16.0 | nM | 7.80 |
| CHEMBL4299655 | — | EC50 | = | 21.0 | nM | 7.68 |
| CHEMBL3823755 | — | EC50 | = | 32.0 | nM | 7.50 |
| CHEMBL3822625 | — | EC50 | = | 39.0 | nM | 7.41 |
| CHEMBL3824159 | — | EC50 | = | 40.0 | nM | 7.40 |
| CHEMBL3823411 | — | EC50 | = | 45.0 | nM | 7.35 |
| CHEMBL3822981 | — | EC50 | = | 56.0 | nM | 7.25 |
| CHEMBL3823448 | — | EC50 | = | 60.0 | nM | 7.22 |
| CHEMBL3823334 | — | EC50 | = | 70.0 | nM | 7.16 |
| CHEMBL3823889 | — | EC50 | = | 80.0 | nM | 7.10 |
| CHEMBL3823221 | — | EC50 | = | 83.0 | nM | 7.08 |
| CHEMBL3823421 | — | EC50 | = | 90.0 | nM | 7.05 |
| CHEMBL3822975 | — | EC50 | = | 100.0 | nM | 7.00 |
| CHEMBL3823878 | — | EC50 | = | 110.0 | nM | 6.96 |
| CHEMBL3823876 | — | EC50 | = | 120.0 | nM | 6.92 |
| CHEMBL3823835 | — | EC50 | = | 130.0 | nM | 6.89 |
| CHEMBL3823333 | — | EC50 | = | 180.0 | nM | 6.75 |
| CHEMBL3823760 | — | EC50 | = | 300.0 | nM | 6.52 |
| CHEMBL2177395 | — | EC50 | = | 520.0 | nM | 6.28 |
| CHEMBL3824332 | — | EC50 | > | 1000.0 | nM | - |
| CHEMBL3823043 | — | EC50 | > | 1000.0 | nM | - |
| CHEMBL3824079 | — | EC50 | > | 1000.0 | nM | - |
| CHEMBL3824232 | — | EC50 | > | 1000.0 | nM | - |
| CHEMBL3823082 | — | EC50 | > | 1000.0 | nM | - |
| CHEMBL3823541 | — | EC50 | > | 1000.0 | nM | - |
| CHEMBL3823133 | — | EC50 | > | 1000.0 | nM | - |
| CHEMBL3823291 | — | EC50 | > | 1000.0 | nM | - |
| CHEMBL3824241 | — | EC50 | > | 1000.0 | nM | - |
| CHEMBL3823722 | — | EC50 | > | 1000.0 | nM | - |
| CHEMBL3822888 | — | EC50 | > | 1000.0 | nM | - |
| CHEMBL4299689 | — | EC50 | > | 1000.0 | nM | - |
| CHEMBL3823994 | — | EC50 | > | 1000.0 | nM | - |
| CHEMBL4299648 | — | EC50 | > | 1000.0 | nM | - |
| CHEMBL4299622 | — | EC50 | > | 1000.0 | nM | - |
| CHEMBL3823847 | — | EC50 | > | 1000.0 | nM | - |
| CHEMBL3823327 | — | EC50 | > | 1000.0 | nM | - |
| CHEMBL3823985 | — | EC50 | > | 1000.0 | nM | - |
| CHEMBL3823144 | — | EC50 | > | 1000.0 | nM | - |
| CHEMBL3822792 | — | EC50 | > | 1000.0 | nM | - |
| CHEMBL3823976 | — | EC50 | > | 1000.0 | nM | - |
| CHEMBL3822459 | — | EC50 | > | 1000.0 | nM | - |
| CHEMBL4299662 | — | EC50 | > | 1000.0 | nM | - |
| CHEMBL3823643 | — | EC50 | > | 1000.0 | nM | - |
| CHEMBL3824278 | — | EC50 | > | 1000.0 | nM | - |
| CHEMBL3822928 | — | EC50 | > | 1000.0 | nM | - |
| CHEMBL4299631 | — | EC50 | > | 1000.0 | nM | - |
| CHEMBL3822636 | — | EC50 | > | 1000.0 | nM | - |