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Assay Detail

CHEMBL3829095

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of recombinant human DHFR assessed as reduction in NADPH oxidation using dihydrofolate as substrate preincubated for 5 mins followed by substrate addition
9
Total Activities
9
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Dihydrofolate reductase (CHEMBL202)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Charged Nonclassical Antifolates with Activity Against Gram-Positive and Gram-Negative Pathogens.
Scocchera E, Reeve SM, Keshipeddy S, Lombardo MN, Hajian B, Sochia AE, Alverson JB, Priestley ND, Anderson AC, Wright DL.
ACS Med Chem Lett (2016) 7 : 692 -696
PubMed 27437079 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 9 6.19 6.80

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL3828291 1 6.80
CHEMBL3827532 1 6.70
CHEMBL3828485 1 6.63
CHEMBL3828724 1 6.46
CHEMBL3827326 1 6.42
CHEMBL3828581 1 6.41
CHEMBL3827760 1 6.35
CHEMBL3827086 1 5.60
CHEMBL22 TRIMETHOPRIM 4.0 1 4.34

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL3828291 Ki = 158.77 nM 6.80
CHEMBL3827532 Ki = 200.77 nM 6.70
CHEMBL3828485 Ki = 234.23 nM 6.63
CHEMBL3828724 Ki = 346.15 nM 6.46
CHEMBL3827326 Ki = 376.62 nM 6.42
CHEMBL3828581 Ki = 388.62 nM 6.41
CHEMBL3827760 Ki = 451.15 nM 6.35
CHEMBL3827086 Ki = 2494.9 nM 5.60
CHEMBL22 TRIMETHOPRIM Ki = 45783.5 nM 4.34