Assay Detail
Functional
CHEMBL3832791
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AntiLeishmania activity L. donovani (macrophages) IC50 (uM)
14
Total Activities
14
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Leishmania donovani |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
MMV Pathogen Box Bioactivity Data
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 14 | 5.06 | 5.58 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL472881 | — | — | 1 | 5.58 |
| CHEMBL474899 | — | — | 1 | 5.38 |
| CHEMBL511692 | — | — | 1 | 5.29 |
| CHEMBL1683021 | — | — | 1 | 4.89 |
| CHEMBL1094051 | — | — | 1 | 4.65 |
| CHEMBL394474 | — | — | 1 | 4.58 |
| CHEMBL394241 | — | — | 1 | - |
| CHEMBL1683016 | — | — | 1 | - |
| CHEMBL458799 | — | — | 1 | - |
| CHEMBL472854 | — | — | 1 | - |
| CHEMBL3637892 | — | — | 1 | - |
| CHEMBL1197563 | — | — | 1 | - |
| CHEMBL519040 | — | — | 1 | - |
| CHEMBL241634 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL472881 | — | IC50 | = | 2600.0 | nM | 5.58 |
| CHEMBL474899 | — | IC50 | = | 4200.0 | nM | 5.38 |
| CHEMBL511692 | — | IC50 | = | 5170.0 | nM | 5.29 |
| CHEMBL1683021 | — | IC50 | = | 12800.0 | nM | 4.89 |
| CHEMBL1094051 | — | IC50 | = | 22200.0 | nM | 4.65 |
| CHEMBL394474 | — | IC50 | = | 26100.0 | nM | 4.58 |
| CHEMBL394241 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL1683016 | — | IC50 | > | 30000.0 | nM | - |
| CHEMBL458799 | — | IC50 | > | 30000.0 | nM | - |
| CHEMBL472854 | — | IC50 | > | 30000.0 | nM | - |
| CHEMBL3637892 | — | IC50 | > | 30000.0 | nM | - |
| CHEMBL1197563 | — | IC50 | > | 30000.0 | nM | - |
| CHEMBL519040 | — | IC50 | > | 30000.0 | nM | - |
| CHEMBL241634 | — | IC50 | > | 30000.0 | nM | - |