Assay Detail
Binding
CHEMBL3853648
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Activity at NET in rat synaptosomes obtained from whole brain minus striatum and cerebellum assessed as release of [3H]MPP+ by liquid scintillation counting method
13
Total Activities
13
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Rattus norvegicus |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 13 | 6.67 | 8.15 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL612 | DEXTROAMPHETAMINE | 4.0 | 1 | 8.15 |
| CHEMBL471839 | — | — | 1 | 7.96 |
| CHEMBL3921422 | — | — | 1 | 6.86 |
| CHEMBL3963971 | — | — | 1 | 6.77 |
| CHEMBL3896023 | — | — | 1 | 6.68 |
| CHEMBL3982376 | — | — | 1 | 6.62 |
| CHEMBL3913053 | — | — | 1 | 6.55 |
| CHEMBL3965276 | — | — | 1 | 6.52 |
| CHEMBL3933915 | — | — | 1 | 6.51 |
| CHEMBL3912463 | — | — | 1 | 6.30 |
| CHEMBL3930376 | — | — | 1 | 6.21 |
| CHEMBL3974905 | — | — | 1 | 6.11 |
| CHEMBL3945529 | — | — | 1 | 5.53 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL612 | DEXTROAMPHETAMINE | EC50 | = | 7.1 | nM | 8.15 |
| CHEMBL471839 | — | EC50 | = | 11.1 | nM | 7.96 |
| CHEMBL3921422 | — | EC50 | = | 138.0 | nM | 6.86 |
| CHEMBL3963971 | — | EC50 | = | 170.0 | nM | 6.77 |
| CHEMBL3896023 | — | EC50 | = | 211.0 | nM | 6.68 |
| CHEMBL3982376 | — | EC50 | = | 239.0 | nM | 6.62 |
| CHEMBL3913053 | — | EC50 | = | 279.0 | nM | 6.55 |
| CHEMBL3965276 | — | EC50 | = | 301.0 | nM | 6.52 |
| CHEMBL3933915 | — | EC50 | = | 308.0 | nM | 6.51 |
| CHEMBL3912463 | — | EC50 | = | 496.0 | nM | 6.30 |
| CHEMBL3930376 | — | EC50 | = | 621.0 | nM | 6.21 |
| CHEMBL3974905 | — | EC50 | = | 784.0 | nM | 6.11 |
| CHEMBL3945529 | — | EC50 | = | 2980.0 | nM | 5.53 |