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Assay Detail

CHEMBL3853654

Review assay metadata, readout intent, target linkage, and publication context from the same page.

ADMET
Agonist activity at human 5-HT2A receptor expressed in HEK293 cells by [3H]-inositol phosphate accumulation assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type ADMET
Organism Homo sapiens
Cell Type HEK293
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

5-hydroxytryptamine receptor 2A (CHEMBL224)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Medchemcomm (2016) 7 : 1657 -1663
· DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 1 6.33 6.33

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL471839 1 6.33

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL471839 EC50 = 466.0 nM 6.33