Assay Detail
Binding
CHEMBL3857901
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of glutamate transporter (unknown origin) assessed as suppression of synaptosomal uptake of L-glutamate
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Polycyclic Polyprenylated Acylphloroglucinol Congeners from Hypericum scabrum.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 5.70 | 5.70 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1237210 | — | — | 1 | 5.70 |
| CHEMBL536352 | — | — | 1 | 5.70 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1237210 | — | IC50 | = | 2000.0 | nM | 5.70 |
| CHEMBL536352 | — | IC50 | = | 2000.0 | nM | 5.70 |