Assay Detail
Binding
CHEMBL3869434
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Inhibition of Penicillium decumbens alpha-L-rhamnosidase
7
Total Activities
7
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Penicillium decumbens |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Strategy for designing selective α-l-rhamnosidase inhibitors: Synthesis and biological evaluation of l-DMDP cyclic isothioureas.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 7 | 5.45 | 7.50 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL596461 | — | — | 1 | 7.50 |
| CHEMBL3913830 | — | — | 1 | 5.48 |
| CHEMBL608711 | — | — | 1 | 5.43 |
| CHEMBL593715 | — | — | 1 | 5.30 |
| CHEMBL1169558 | — | — | 1 | 4.68 |
| CHEMBL3984167 | — | — | 1 | 4.28 |
| CHEMBL3955539 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL596461 | — | IC50 | = | 32.0 | nM | 7.50 |
| CHEMBL3913830 | — | IC50 | = | 3300.0 | nM | 5.48 |
| CHEMBL608711 | — | IC50 | = | 3700.0 | nM | 5.43 |
| CHEMBL593715 | — | IC50 | = | 5000.0 | nM | 5.30 |
| CHEMBL1169558 | — | IC50 | = | 21000.0 | nM | 4.68 |
| CHEMBL3984167 | — | IC50 | = | 52800.0 | nM | 4.28 |
| CHEMBL3955539 | — | IC50 | = | 850000.0 | nM | - |