Assay Detail
Binding
CHEMBL3876376
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Displacement of [125I]peptide YY from Y2 receptor in human KAN-TS cells measured after 60 mins by scintillation counting method
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Cell Type | KAN-TS |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Structure-anticonvulsant activity studies in the group of (E)-N-cinnamoyl aminoalkanols derivatives monosubstituted in phenyl ring with 4-Cl, 4-CH3 or 2-CH3.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 10.55 | 10.55 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL438945 | HUMAN NEUROPEPTIDE Y | 1.0 | 1 | 10.55 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL438945 | HUMAN NEUROPEPTIDE Y | IC50 | = | 0.028 | nM | 10.55 |