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Assay Detail

CHEMBL3880957

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Potentiation of chloroquine-induced anitiparasitic activity in chloroquine-resistant/verapamil-sensitive Plasmodium falciparum FCB assessed as chloroquine IC50 (Rvb = 325 nM)
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Plasmodium falciparum
Confidence 1 — Organism
Curated By Autocuration

Target

Plasmodium falciparum (CHEMBL364)
Type ORGANISM
Organism Plasmodium falciparum

Publication

Isoform Selective HDAC Inhibitors
(2010)

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 7.22 7.22

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL227120 1 7.22

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL227120 IC50 = 60.0 nM 7.22