Assay Detail
Binding
CHEMBL3883095
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Displacement of [3H]PGE2 from from human EP4 receptor expressed in HEK293 cells membranes incubated for 60 mins
30
Total Activities
30
Compounds Tested
2
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Cell Type | HEK293 |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Prostaglandin E2 receptor EP4 subtype (CHEMBL1836) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Therapeutic compounds
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 27 | 5.17 | 5.85 |
| IC50 | 3 | 4.88 | 4.88 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3936540 | — | — | 1 | 5.85 |
| CHEMBL3959926 | — | — | 1 | 5.63 |
| CHEMBL3959653 | — | — | 1 | 5.55 |
| CHEMBL3901873 | — | — | 1 | 5.06 |
| CHEMBL3939358 | — | — | 1 | 4.88 |
| CHEMBL1722929 | — | — | 1 | 4.82 |
| CHEMBL3922151 | — | — | 1 | 4.82 |
| CHEMBL3920796 | — | — | 1 | 4.82 |
| CHEMBL3918084 | — | — | 1 | 4.82 |
| CHEMBL3920756 | — | — | 1 | - |
| CHEMBL3909754 | — | — | 1 | - |
| CHEMBL3959769 | — | — | 1 | - |
| CHEMBL3908484 | — | — | 1 | - |
| CHEMBL3929446 | — | — | 1 | - |
| CHEMBL3928130 | — | — | 1 | - |
| CHEMBL3905811 | — | — | 1 | - |
| CHEMBL3906402 | — | — | 1 | - |
| CHEMBL3973347 | — | — | 1 | - |
| CHEMBL3971632 | — | — | 1 | - |
| CHEMBL3921784 | — | — | 1 | - |
| CHEMBL3986829 | — | — | 1 | - |
| CHEMBL3934202 | — | — | 1 | - |
| CHEMBL3924987 | — | — | 1 | - |
| CHEMBL3975238 | — | — | 1 | - |
| CHEMBL3977724 | — | — | 1 | - |
| CHEMBL3907809 | — | — | 1 | - |
| CHEMBL3918349 | — | — | 1 | - |
| CHEMBL3915040 | — | — | 1 | - |
| CHEMBL3891401 | — | — | 1 | - |
| CHEMBL3892847 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3936540 | — | Ki | = | 1400.0 | nM | 5.85 |
| CHEMBL3959926 | — | Ki | = | 2364.0 | nM | 5.63 |
| CHEMBL3959653 | — | Ki | = | 2809.0 | nM | 5.55 |
| CHEMBL3901873 | — | Ki | = | 8752.0 | nM | 5.06 |
| CHEMBL3939358 | — | IC50 | = | 13100.0 | nM | 4.88 |
| CHEMBL1722929 | — | Ki | = | 15000.0 | nM | 4.82 |
| CHEMBL3922151 | — | Ki | = | 15000.0 | nM | 4.82 |
| CHEMBL3920796 | — | Ki | = | 15000.0 | nM | 4.82 |
| CHEMBL3918084 | — | Ki | = | 15000.0 | nM | 4.82 |
| CHEMBL3920756 | — | Ki | > | 10000.0 | nM | - |
| CHEMBL3909754 | — | Ki | > | 10000.0 | nM | - |
| CHEMBL3959769 | — | Ki | > | 10000.0 | nM | - |
| CHEMBL3908484 | — | Ki | > | 10000.0 | nM | - |
| CHEMBL3929446 | — | Ki | > | 10000.0 | nM | - |
| CHEMBL3928130 | — | Ki | > | 10000.0 | nM | - |
| CHEMBL3905811 | — | Ki | > | 10000.0 | nM | - |
| CHEMBL3906402 | — | Ki | > | 10000.0 | nM | - |
| CHEMBL3973347 | — | Ki | > | 10000.0 | nM | - |
| CHEMBL3971632 | — | Ki | >= | 3842.0 | nM | - |
| CHEMBL3921784 | — | Ki | > | 10000.0 | nM | - |
| CHEMBL3986829 | — | IC50 | - | — | - | |
| CHEMBL3934202 | — | IC50 | - | — | - | |
| CHEMBL3924987 | — | Ki | > | 10000.0 | nM | - |
| CHEMBL3975238 | — | Ki | > | 10000.0 | nM | - |
| CHEMBL3977724 | — | Ki | >= | 3288.0 | nM | - |
| CHEMBL3907809 | — | Ki | > | 10000.0 | nM | - |
| CHEMBL3918349 | — | Ki | > | 10000.0 | nM | - |
| CHEMBL3915040 | — | Ki | > | 10000.0 | nM | - |
| CHEMBL3891401 | — | Ki | > | 10000.0 | nM | - |
| CHEMBL3892847 | — | Ki | >= | 6032.0 | nM | - |