Assay Detail

CHEMBL3889032

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Binding

Inhibition Assay: Inhibition of recombinant FGFR-2 tyrosine kinase using exogenous substrate.

ChEMBL ↗

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Target

Fibroblast growth factor receptor 2 (CHEMBL4142) ↗

Open DB target context

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Fibroblast growth factor receptor 2 (CHEMBL4142) is the working anchor for this assay review. Loading the live Open DB target snapshot…

Primary target Fibroblast growth factor receptor 2

CHEMBL4142

Anchored from Assay target.

Protein identity Fibroblast growth factor receptor 2

Disease frame Disease evidence pending

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Review focus Open DB context pending

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Total Activities

Compounds Tested

Activity Types

Assay Parameters

Assay Information

Assay Type	Binding
Organism	Homo sapiens
Confidence	8 — Homologous single protein target
Curated By	Autocuration

Target

Fibroblast growth factor receptor 2 (CHEMBL4142) ↗

Type	SINGLE PROTEIN
Organism	Homo sapiens

Publication

Ocular formulations for drug-delivery to the posterior segment of the eye

(2016)

Activity Statistics

Type	Count	Avg pChEMBL	Best pChEMBL
IC50	1	8.06	8.06

Compounds Tested

Compound	Name	Phase	Activities	Best pChEMBL
CHEMBL253969	OSI-632	2.0	1	8.06

Activity Data

Compound	Name	Type	Rel.	Value	Units	pChEMBL
CHEMBL253969	OSI-632	IC50	=	8.79	nM	8.06