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Assay Detail

CHEMBL3999028

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of PI4K3beta (unknown origin) by select screen kinase profiling assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

Unchecked (CHEMBL612545)
Type UNCHECKED

Publication

Discovery of Multitarget Agents Active as Broad-Spectrum Antivirals and Correctors of Cystic Fibrosis Transmembrane Conductance Regulator for Associated Pulmonary Diseases.
Tassini S, Sun L, Lanko K, Crespan E, Langron E, Falchi F, Kissova M, Armijos-Rivera JI, Delang L, Mirabelli C, Neyts J, Pieroni M, Cavalli A, Costantino G, Maga G, Vergani P, Leyssen P, Radi M.
J Med Chem (2017) 60 : 1400 -1416
PubMed 28122178 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 7.22 7.22

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL2397317 1 7.22

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL2397317 IC50 = 60.0 nM 7.22