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Assay Detail

CHEMBL4007597

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of alpha-hexosaminidase (unknown origin)
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Beta-hexosaminidase subunit alpha (CHEMBL1250415)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

(5aR)-5a-C-Pentyl-4-epi-isofagomine: A powerful inhibitor of lysosomal β-galactosidase and a remarkable chaperone for mutations associated with GM1-gangliosidosis and Morquio disease type B.
Front S, Biela-Banaś A, Burda P, Ballhausen D, Higaki K, Caciotti A, Morrone A, Charollais-Thoenig J, Gallienne E, Demotz S, Martin OR.
Eur J Med Chem (2017) 126 : 160 -170
PubMed 27750150 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 7.00 7.00

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL4097052 1 7.00

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4097052 IC50 = 100.0 nM 7.00