Assay Detail
Functional
CHEMBL4012795
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Antiviral activity against Human rhinovirus B14 infected in human H1HeLa cells assessed as protection against virus induced cytopathic effect after 3 days by MTT assay
43
Total Activities
43
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | rhinovirus B14 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
A Novel Series of Highly Potent Small Molecule Inhibitors of Rhinovirus Replication.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 43 | 5.57 | 7.51 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2062774 | VAPENDAVIR | 2.0 | 1 | 7.51 |
| CHEMBL141157 | IMOCITRELVIR | 2.0 | 1 | 7.35 |
| CHEMBL4086772 | — | — | 1 | 7.16 |
| CHEMBL29609 | PLECONARIL | 2.0 | 1 | 7.12 |
| CHEMBL4062307 | — | — | 1 | 6.09 |
| CHEMBL4095440 | — | — | 1 | 5.77 |
| CHEMBL4105623 | — | — | 1 | 5.77 |
| CHEMBL4086764 | — | — | 1 | 5.75 |
| CHEMBL4084999 | — | — | 1 | 5.72 |
| CHEMBL4065340 | — | — | 1 | 5.70 |
| CHEMBL4073941 | — | — | 1 | 5.68 |
| CHEMBL4068042 | — | — | 1 | 5.68 |
| CHEMBL4103195 | — | — | 1 | 5.54 |
| CHEMBL4059561 | — | — | 1 | 5.47 |
| CHEMBL4078916 | — | — | 1 | 5.00 |
| CHEMBL4094501 | — | — | 1 | 4.96 |
| CHEMBL4073774 | — | — | 1 | 4.93 |
| CHEMBL4100582 | — | — | 1 | 4.91 |
| CHEMBL4068049 | — | — | 1 | 4.87 |
| CHEMBL4087372 | — | — | 1 | 4.61 |
| CHEMBL4095433 | — | — | 1 | 4.25 |
| CHEMBL4098020 | — | — | 1 | 4.16 |
| CHEMBL4081621 | — | — | 1 | 4.08 |
| CHEMBL4080676 | — | — | 1 | - |
| CHEMBL4063354 | — | — | 1 | - |
| CHEMBL4090314 | — | — | 1 | - |
| CHEMBL4065333 | — | — | 1 | - |
| CHEMBL4078907 | — | — | 1 | - |
| CHEMBL4103185 | — | — | 1 | - |
| CHEMBL4100479 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2062774 | VAPENDAVIR | EC50 | = | 31.0 | nM | 7.51 |
| CHEMBL141157 | IMOCITRELVIR | EC50 | = | 45.0 | nM | 7.35 |
| CHEMBL4086772 | — | EC50 | = | 70.0 | nM | 7.16 |
| CHEMBL29609 | PLECONARIL | EC50 | = | 75.0 | nM | 7.12 |
| CHEMBL4062307 | — | EC50 | = | 820.0 | nM | 6.09 |
| CHEMBL4095440 | — | EC50 | = | 1700.0 | nM | 5.77 |
| CHEMBL4105623 | — | EC50 | = | 1700.0 | nM | 5.77 |
| CHEMBL4086764 | — | EC50 | = | 1800.0 | nM | 5.75 |
| CHEMBL4084999 | — | EC50 | = | 1900.0 | nM | 5.72 |
| CHEMBL4065340 | — | EC50 | = | 2000.0 | nM | 5.70 |
| CHEMBL4073941 | — | EC50 | = | 2100.0 | nM | 5.68 |
| CHEMBL4068042 | — | EC50 | = | 2100.0 | nM | 5.68 |
| CHEMBL4103195 | — | EC50 | = | 2900.0 | nM | 5.54 |
| CHEMBL4059561 | — | EC50 | = | 3400.0 | nM | 5.47 |
| CHEMBL4078916 | — | EC50 | = | 10100.0 | nM | 5.00 |
| CHEMBL4094501 | — | EC50 | = | 11000.0 | nM | 4.96 |
| CHEMBL4073774 | — | EC50 | = | 11700.0 | nM | 4.93 |
| CHEMBL4100582 | — | EC50 | = | 12400.0 | nM | 4.91 |
| CHEMBL4068049 | — | EC50 | = | 13500.0 | nM | 4.87 |
| CHEMBL4087372 | — | EC50 | = | 24600.0 | nM | 4.61 |
| CHEMBL4095433 | — | EC50 | = | 56600.0 | nM | 4.25 |
| CHEMBL4098020 | — | EC50 | = | 68600.0 | nM | 4.16 |
| CHEMBL4081621 | — | EC50 | = | 82500.0 | nM | 4.08 |
| CHEMBL4070927 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL1235858 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL4087741 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL4084280 | — | EC50 | > | 18800.0 | nM | - |
| CHEMBL4102246 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL4091888 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL4071055 | — | EC50 | > | 42500.0 | nM | - |
| CHEMBL4099621 | — | EC50 | > | 110.0 | nM | - |
| CHEMBL4084131 | — | EC50 | > | 52300.0 | nM | - |
| CHEMBL4062420 | — | EC50 | > | 70900.0 | nM | - |
| CHEMBL4104906 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL4081513 | — | EC50 | > | 42400.0 | nM | - |
| CHEMBL4082467 | — | EC50 | > | 24900.0 | nM | - |
| CHEMBL4100479 | — | EC50 | > | 7600.0 | nM | - |
| CHEMBL4103185 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL4078907 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL4065333 | — | EC50 | > | 16000.0 | nM | - |
| CHEMBL4090314 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL4063354 | — | EC50 | > | 14600.0 | nM | - |
| CHEMBL4080676 | — | EC50 | > | 82000.0 | nM | - |