Assay Detail
Functional
CHEMBL4012802
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Antiviral activity against Human poliovirus 3 infected in human HeLa cells assessed as protection against virus induced cytopathic effect after 2 days by MTT assay
41
Total Activities
41
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Poliovirus 3 |
| Cell Type | HeLa |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
A Novel Series of Highly Potent Small Molecule Inhibitors of Rhinovirus Replication.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 41 | 6.10 | 8.02 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4073941 | — | — | 1 | 8.02 |
| CHEMBL4086764 | — | — | 1 | 8.00 |
| CHEMBL4094501 | — | — | 1 | 7.36 |
| CHEMBL4086772 | — | — | 1 | 7.20 |
| CHEMBL4084999 | — | — | 1 | 7.15 |
| CHEMBL4063354 | — | — | 1 | 7.14 |
| CHEMBL1235858 | — | — | 1 | 7.10 |
| CHEMBL4065340 | — | — | 1 | 7.06 |
| CHEMBL4095440 | — | — | 1 | 7.03 |
| CHEMBL4103185 | — | — | 1 | 6.75 |
| CHEMBL4084280 | — | — | 1 | 6.47 |
| CHEMBL4065333 | — | — | 1 | 6.46 |
| CHEMBL4059561 | — | — | 1 | 6.42 |
| CHEMBL4068042 | — | — | 1 | 6.39 |
| CHEMBL4103195 | — | — | 1 | 6.15 |
| CHEMBL29609 | PLECONARIL | 2.0 | 1 | 5.85 |
| CHEMBL4104906 | — | — | 1 | 5.75 |
| CHEMBL4095433 | — | — | 1 | 5.72 |
| CHEMBL4078916 | — | — | 1 | 5.70 |
| CHEMBL4105623 | — | — | 1 | 5.19 |
| CHEMBL4062307 | — | — | 1 | 5.04 |
| CHEMBL4080676 | — | — | 1 | 5.03 |
| CHEMBL4062420 | — | — | 1 | 4.88 |
| CHEMBL4081621 | — | — | 1 | 4.26 |
| CHEMBL4100582 | — | — | 1 | 4.23 |
| CHEMBL4078907 | — | — | 1 | 4.22 |
| CHEMBL4087372 | — | — | 1 | 4.19 |
| CHEMBL4090314 | — | — | 1 | - |
| CHEMBL4068049 | — | — | 1 | - |
| CHEMBL4087741 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4073941 | — | EC50 | = | 9.5 | nM | 8.02 |
| CHEMBL4086764 | — | EC50 | = | 10.0 | nM | 8.00 |
| CHEMBL4094501 | — | EC50 | = | 44.0 | nM | 7.36 |
| CHEMBL4086772 | — | EC50 | = | 63.0 | nM | 7.20 |
| CHEMBL4084999 | — | EC50 | = | 71.0 | nM | 7.15 |
| CHEMBL4063354 | — | EC50 | = | 72.0 | nM | 7.14 |
| CHEMBL1235858 | — | EC50 | = | 80.0 | nM | 7.10 |
| CHEMBL4065340 | — | EC50 | = | 87.0 | nM | 7.06 |
| CHEMBL4095440 | — | EC50 | = | 93.0 | nM | 7.03 |
| CHEMBL4103185 | — | EC50 | = | 180.0 | nM | 6.75 |
| CHEMBL4084280 | — | EC50 | = | 340.0 | nM | 6.47 |
| CHEMBL4065333 | — | EC50 | = | 350.0 | nM | 6.46 |
| CHEMBL4059561 | — | EC50 | = | 380.0 | nM | 6.42 |
| CHEMBL4068042 | — | EC50 | = | 410.0 | nM | 6.39 |
| CHEMBL4103195 | — | EC50 | = | 710.0 | nM | 6.15 |
| CHEMBL29609 | PLECONARIL | EC50 | = | 1400.0 | nM | 5.85 |
| CHEMBL4104906 | — | EC50 | = | 1800.0 | nM | 5.75 |
| CHEMBL4095433 | — | EC50 | = | 1900.0 | nM | 5.72 |
| CHEMBL4078916 | — | EC50 | = | 2000.0 | nM | 5.70 |
| CHEMBL4105623 | — | EC50 | = | 6400.0 | nM | 5.19 |
| CHEMBL4062307 | — | EC50 | = | 9100.0 | nM | 5.04 |
| CHEMBL4080676 | — | EC50 | = | 9400.0 | nM | 5.03 |
| CHEMBL4062420 | — | EC50 | = | 13100.0 | nM | 4.88 |
| CHEMBL4081621 | — | EC50 | = | 55400.0 | nM | 4.26 |
| CHEMBL4100582 | — | EC50 | = | 58700.0 | nM | 4.23 |
| CHEMBL4078907 | — | EC50 | = | 60100.0 | nM | 4.22 |
| CHEMBL4087372 | — | EC50 | = | 64300.0 | nM | 4.19 |
| CHEMBL4084131 | — | EC50 | > | 46900.0 | nM | - |
| CHEMBL4073774 | — | EC50 | > | 45600.0 | nM | - |
| CHEMBL4098020 | — | EC50 | > | 90100.0 | nM | - |
| CHEMBL4070927 | — | EC50 | > | 47600.0 | nM | - |
| CHEMBL4081513 | — | EC50 | > | 43900.0 | nM | - |
| CHEMBL4082467 | — | EC50 | > | 26200.0 | nM | - |
| CHEMBL4100479 | — | EC50 | > | 12900.0 | nM | - |
| CHEMBL4099621 | — | EC50 | > | 450.0 | nM | - |
| CHEMBL4071055 | — | EC50 | > | 44400.0 | nM | - |
| CHEMBL4091888 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL4102246 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL4087741 | — | EC50 | > | 68300.0 | nM | - |
| CHEMBL4068049 | — | EC50 | > | 16700.0 | nM | - |
| CHEMBL4090314 | — | EC50 | > | 100000.0 | nM | - |