Assay Detail
Binding
CHEMBL4014605
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Binding affinity to RXR (unknown origin)
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Opportunities and Challenges for Fatty Acid Mimetics in Drug Discovery.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Kd | 3 | 6.02 | 8.05 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL705 | ALITRETINOIN | 4.0 | 1 | 8.05 |
| CHEMBL367149 | DOCONEXENT | 3.0 | 1 | 5.00 |
| CHEMBL8659 | OLEIC ACID | 2.0 | 1 | 5.00 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL705 | ALITRETINOIN | Kd | = | 9.0 | nM | 8.05 |
| CHEMBL367149 | DOCONEXENT | Kd | = | 10000.0 | nM | 5.00 |
| CHEMBL8659 | OLEIC ACID | Kd | = | 10000.0 | nM | 5.00 |