Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL4014613

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Displacement of [3H]LTD4 from cysteinyl leukotriene receptor (unknown origin) after 60 mins
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

Unchecked (CHEMBL612545)
Type UNCHECKED

Publication

Opportunities and Challenges for Fatty Acid Mimetics in Drug Discovery.
Proschak E, Heitel P, Kalinowsky L, Merk D.
J Med Chem (2017) 60 : 5235 -5266
PubMed 28252961 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 5.22 5.22

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL127905 1 5.22

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL127905 IC50 = 6000.0 nM 5.22