Assay Detail
Binding
CHEMBL4014619
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of cysteinyl leukotriene receptor in guinea pig trachea strip assessed as inhibition of LTD4-induced trachea strip contraction preincubated for 2 mins followed by LTD4 induction
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Cavia porcellus |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Opportunities and Challenges for Fatty Acid Mimetics in Drug Discovery.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 5.05 | 5.05 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL173443 | — | — | 1 | 5.05 |
| CHEMBL173278 | — | — | 1 | 5.05 |
| CHEMBL174471 | — | — | 1 | 5.05 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL173443 | — | IC50 | = | 9000.0 | nM | 5.05 |
| CHEMBL173278 | — | IC50 | = | 9000.0 | nM | 5.05 |
| CHEMBL174471 | — | IC50 | = | 9000.0 | nM | 5.05 |