Assay Detail
Binding
CHEMBL4019778
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Binding affinity to human TRPV1 expressed in CHO cells after 45 mins by scintillation counting method
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Transient receptor potential cation channel subfamily V member 1 (CHEMBL4794) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Novel Radiolabeled Vanilloid with Enhanced Specificity for Human Transient Receptor Potential Vanilloid 1 (TRPV1).
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Kd | 3 | 9.12 | 9.23 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4095861 | — | — | 1 | 9.23 |
| CHEMBL4077829 | — | — | 1 | 9.23 |
| CHEMBL4060041 | — | — | 1 | 8.91 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4095861 | — | Kd | = | 0.589 | nM | 9.23 |
| CHEMBL4077829 | — | Kd | = | 0.59 | nM | 9.23 |
| CHEMBL4060041 | — | Kd | = | 1.23 | nM | 8.91 |